Angiotensin converting enzyme inhibitors for long-term management of acute coronary syndromes
Angiotensin converting enzyme inhibitors (ACEIs) reduce cardiovascular mortality after myocardial infarction. Unless contraindicated, start an ACEI within 24 to 48 hours of acute myocardial infarction.
Contraindications to early ACEI use include haemodynamic instability and hypotension (systolic pressure less than 90 mmHg).
Suitable ACEI regimens for long-term management of acute coronary syndromes are1:
1captopril 6.25 mg orally, twice daily, increasing to maximum 150 mg daily in divided doses captopril captopril captopril
OR
1enalapril 2.5 mg orally, daily, increasing to maximum 40 mg daily enalapril enalapril enalapril
OR
1fosinopril 5 mg orally, daily, increasing to maximum 40 mg daily fosinopril fosinopril fosinopril
OR
1lisinopril 2.5 mg orally, daily, increasing to maximum 40 mg daily lisinopril lisinopril lisinopril
OR
1perindopril arginine 2.5 mg orally, daily, increasing to maximum 10 mg daily perindopril perindopril perindopril
OR
1perindopril erbumine 2 mg orally, daily, increasing to maximum 8 mg daily perindopril perindopril perindopril
OR
1quinapril 2.5 mg orally, daily, increasing to maximum 40 mg daily quinapril quinapril quinapril
OR
1ramipril 2.5 mg orally, daily, increasing to maximum 10 mg daily ramipril ramipril ramipril
OR
1trandolapril 0.5 mg orally, daily, increasing to maximum 4 mg daily2. trandolapril trandolapril trandolapril
Titrate to the maximum tolerated dose and continue the ACEI long term. Gradually increase the dose within 4 to 6 weeks after discharge. Monitor for hypotension, kidney impairment and hyperkalaemia.
In patients with clinical heart failure and a left ventricular ejection fraction (LVEF) of 40% or less, an alternative renin-angiotensin system inhibitor (eg sacubitril+valsartan) may be indicated instead of an ACEI; for more information, see Renin-angiotensin system inhibitors for HFrEF.
The combination of an ACEI with an angiotensin II receptor blocker (ARB) is not recommended except with specialist advice.