Immunomodulatory drugs for idiopathic inflammatory myopathies (excluding inclusion body myositis)

Conventional synthetic disease-modifying antirheumatic drugs (csDMARDs) are often used for their corticosteroid-sparing effects and to achieve remission of disease. For idiopathic inflammatory myopathies, the csDMARDs most commonly used are azathioprine, methotrexate, mycophenolate and ciclosporinPipitone, 2020.

The usual dose of azathioprine for idiopathic inflammatory myopathy is:

azathioprine 1.5 to 2.5 mg/kg orally, daily. azathioprine azathioprine azathioprine

For additional considerations specific to azathioprine use, see Specific considerations for use of conventional synthetic disease-modifying antirheumatic drugs (csDMARDs).

The usual dose of methotrexate for idiopathic inflammatory myopathy is:

1methotrexate 10 to 25 mg orally, on one specified day once weekly methotrexate methotrexate methotrexate

OR

1methotrexate 10 to 25 mg subcutaneously, on one specified day once weekly methotrexate methotrexate methotrexate

PLUS with either of the above

folic acid 5 to 10 mg orally, weekly (not on the same day as methotrexate). folic acid folic acid folic acid

For additional considerations specific to methotrexate use, see Specific considerations for use of conventional synthetic disease-modifying antirheumatic drugs (csDMARDs).

The usual doses of mycophenolate for idiopathic inflammatory myopathy are:

1mycophenolate mofetil 500 mg orally, twice daily; increase the dose gradually as tolerated aiming for 1000 to 1500 mg orally, twice daily (maximum 3000 mg daily)1 mycophenolate mofetil mycophenolate mofetil mycophenolate mofetil

OR

1mycophenolate sodium 360 mg orally, twice daily; increase the dose gradually as tolerated to a maximum of 1080 mg orally, twice daily. mycophenolate sodium mycophenolate sodium (mycophenolic acid) mycophenolate sodium (mycophenolic acid)

For additional considerations specific to mycophenolate use, see Specific considerations for use of conventional synthetic disease-modifying antirheumatic drugs (csDMARDs).

The usual dose of ciclosporin for idiopathic inflammatory myopathy is:

ciclosporin 2.5 to 5 mg/kg orally, daily. ciclosporin ciclosporin ciclosporin

For additional considerations specific to ciclosporin use, see Specific considerations for use of conventional synthetic disease-modifying antirheumatic drugs (csDMARDs).

1 Mycophenolate mofetil is the most commonly used preparation, but if tolerance is a problem, mycophenolate sodium (modified-release preparation) can be substituted.Return