Oral drugs for severe, acute nociceptive pain in adults

The oral route of administration for severe, acute nociceptive pain is preferred when prompt analgesia is not required (eg postoperatively when analgesia has been established). Alternative routes of administration should be used if oral absorption is impaired (eg trauma patients). Irrespective of the route of administration used for initial analgesia, oral administration should be used for ongoing analgesia.

For advice on choosing an opioid or the route of administration for severe, acute nociceptive pain, see Approach to managing severe, acute nociceptive pain.

If oral drug regimens are appropriate for severe, acute nociceptive pain due to an acute illness (eg shingles), or following surgery or trauma, as a three-drug regimen, use:

1 paracetamol immediate-release 1 g orally, 4-to 6-hourly. Maximum dose 4 g in 24 hours acute pain, severe (adults receiving oral opioids) paracetamol    

OR

1 paracetamol modified-release 1.33 g orally, 8-hourly. Maximum dose 4 g in 24 hours paracetamol    

PLUS ONE OF THE FOLLOWING NSAIDS

1 celecoxib 100 to 200 mg orally, twice daily acute pain, severe (adults receiving oral opioids) celecoxib    

OR

1 ibuprofen 200 to 400 mg orally, 3 times daily1 acute pain, severe (adults receiving oral opioids) ibuprofen    

OR

1 naproxen 250 to 500 mg orally, twice daily2 acute pain, severe (adults receiving oral opioids) naproxen    

PLUS ONE OF THE FOLLOWING OPIOIDS

1 morphine immediate-release acute pain, severe (adults) morphine    

adults 39 years or younger: 20 to 35 mg orally, 2-hourly if required. Use the lower end of the dose range initially for patients whose opioid requirements have not been established. Consider lower initial doses for cachectic or frail patients

adults 40 to 59 years: 15 to 30 mg orally, 2-hourly if required. Use the lower end of the dose range initially for patients whose opioid requirements have not been established. Consider lower initial doses for cachectic or frail patients

adults 60 to 69 years: 7.5 to 20 mg orally, 2-hourly if required. Use the lower end of the dose range initially for patients whose opioid requirements have not been established. Consider lower initial doses for cachectic or frail patients

adults 70 to 85 years: 7.5 to 10 mg orally, 2-hourly if required. Use the lower end of the dose range initially for patients whose opioid requirements have not been established. Consider lower initial doses for cachectic or frail patients

adults older than 85 years: 3.5 to 7.5 mg orally, 2-hourly if required. Use the lower end of the dose range initially for patients whose opioid requirements have not been established. Consider lower initial doses for cachectic or frail patients

after each dose, wait 1 hour then assess the patient for signs of opioid-induced ventilatory impairment (using sedation score and respiratory rate) and determine whether pain relief is adequate. See Opioid dose titration in hospital for subsequent management, including top-up doses

OR

1 oxycodone immediate-release acute pain, severe (adults) oxycodone    

adults 39 years or younger: 10 to 25 mg orally, 2-hourly if required. Use the lower end of the dose range initially for patients whose opioid requirements have not been established. Consider lower initial doses for cachectic or frail patients

adults 40 to 59 years: 10 to 20 mg orally, 2-hourly if required. Use the lower end of the dose range initially for patients whose opioid requirements have not been established. Consider lower initial doses for cachectic or frail patients

adults 60 to 69 years: 5 to 15 mg orally, 2-hourly if required. Use the lower end of the dose range initially for patients whose opioid requirements have not been established. Consider lower initial doses for cachectic or frail patients

adults 70 to 85 years: 5 to 10 mg orally, 2-hourly if required. Use the lower end of the dose range initially for patients whose opioid requirements have not been established. Consider lower initial doses for cachectic or frail patients

adults older than 85 years: 2.5 to 5 mg orally, 2-hourly if required. Use the lower end of the dose range initially for patients whose opioid requirements have not been established. Consider lower initial doses for cachectic or frail patients

after each dose, wait 1 hour then assess the patient for signs of opioid-induced ventilatory impairment (using sedation score and respiratory rate) and determine whether pain relief is adequate. See Opioid dose titration in hospital for subsequent management, including top-up doses.

1 Avoid ibuprofen in patients at increased risk of bleeding or gastrointestinal toxicity. In these patients, celecoxib is preferred. See Nonsteroidal anti-inflammatory drugs (NSAIDs) in pain management for further advice on adverse effects and contraindications.Return
2 Avoid naproxen in patients at increased risk of bleeding or gastrointestinal toxicity. In these patients, celecoxib is preferred. See Nonsteroidal anti-inflammatory drugs (NSAIDs) in pain management for further advice on adverse effects and contraindications.Return